There is much confusion online as to whether or not Clenbuterol is an anabolic steroid.
It is frequently mentioned alongside bodybuilding steroids and may be used in stacks with other anabolics.
However, Clenbuterol is a stimulant, or sympathomimetic amine, and not an anabolic steroid.
Other drugs in this family are Adderall, Ephedrine, Albuterol and Caffeine.
This is a large category of drugs, and the above drugs, plus Clenbuterol, Norepinephrine, Epinephrine, etc. are similar to each other and can be thought of as cousins or siblings.
Clenbuterol, specifically, uses a few different methods to stimulate the sympathomimetic central nervous system.
It accomplishes this through adrenoreceptors, which are contained within many different tissues in the body.Click here to buy legal Clenbutrol from CrazyBulk online, without a prescription.
Throughout the tissues which contain these receptors, Clen will create different effects when it meets the receptor, according to the type of cells that contain the receptors.
There are about nine different types of andrenoreceptors in the human body. Because of this they are labeled by number and as either Alpha or Beta.
For instance, the body contains receptors known as Beta-1, Beta-2, Beta-3, etc., and the same for Alpha.
The various sympathomimetic and stimulant compounds are different from their siblings and cousins not only in what actions they do, but in how they act upon these various receptors.
Clen in particular is known for how it interacts with Beta-2 receptors. This explains why it is known as a Beta-2 receptor agonist.
How this relates to the fat burning effects of Clenbuterol will be discussed more extensively.
We will also explain more about how the mechanism of action differs from steroids, but point out that there are some anabolic properties of Clen which is why it may be stacked together with other anabolic steroids in a bodybuilding cycle.
However, the primary effects of this stimulant relate to increasing metabolic activity to burn fat as opposed to building muscle.
Despite the fact that Clenbuterol is used mainly to burn fat among those in entertainment and athletic circles, it was first used in medicine for something quite different.
Sympathomimetics and stimulants of all kinds are used in medicine for treating many different medical problems, and most medical conditions that they are used for can be treated with a variety of medicationsin this class.
Clenbuterol has been used for treatment of asthma. It is a primary ingredient in many asthma inhalers, though it isn’t used in the US any longer for this purpose, with Albuterol taking its place.
Clenbuterol is very effective in the treatment of asthma since it activates Beta-2 receptors, particularly those in cells located in the lining of the bronchial tubes.
This causes bronchial dilation in the throat, nose and lungs, so that the airways are expanded. All sympathomimetics have some degree of usage for bronchial dilation.
The human body creates its own neurotransmitters (Norepinephrine and Epinephrine, also known as Noradrenaline and Adrenaline), that also work as sympathomimetic stimulants, but to a much greater degree.
Clenbuterol is also used medically to treat anaphylactic shock, histamine reactions, swellingand allergic reactions, migraine headaches, arrhythmias, cardiovascular slowdown or shock and hypertension.
As mentioned earlier, Clenbuterol works as a Beta-2 agonist since it does work primarily on the body’s Beta-2 receptors.
But it does work with additional receptor sites as well, just not in as significant of a degree, and with less significant results.
For instance, if you compare Ephedrine and Clenbuterol, you will see that while Ephedrine works on a great deal of both Alpha and Beta receptors equally, Clenbuterol mainly affects Beta-2 receptors.
To put it in simple terms, if the receptors were a collection of nails sticking out of a piece of wood, the effect of Clenbuterol is similar to using a small hammer to nail in one nail individually.
In comparison to Ephedrine, which is like hitting all the nails at once with a sledgehammer. This example isn’t perfect, but it is a good summary of the way Clenbuterol works.
We have talked about how Clenbuterol is used in medicine, for bronchodilation, as well as its other medical uses.
We have yet to talk about and explain the main use for Clenbuterol in weight loss: the effect it has on metabolism of fat.
Clenbuterol is known for its minor anabolic function in muscle tissues, with animal research demonstrating a clear anabolic effect on muscle tissue.
However, it is a minor and very mild effect. These studies have shown, and bodybuilder’s, as well as other human users have shown that the anabolic effects of Clenbuterol are minor, if they are even seen at all.
Research looking at the effect of Clenbuterol on rat skeletal muscle tissue showed that it does have a small anabolic effect on animals, however, it must be used for an extended period of time to have these effects.
This means that anyone looking to use Clenbuterol for an anabolic reason will probably be disappointed.
Clenbuterol, when taken with steroids for performance or physique enhancement, must be seen above all as an aid to help you lose fat, and not for anabolic uses, since it is not effective for this.
Also, it is important to note that these slight anabolic effects in animals were seen after giving them doses which would be very dangerous and extreme in humans.
Because of this, many hypothesize that Clenbuterol may not have any anabolic effect on humans at all.
By activating Beta-2 receptors that are in the fat cell membranes, it can activate and begin the metabolism of fat cells directly, beginning the triglyceride breakdown process, in which they are converted into free fatty acids.
The Beta-2 receptors located on fat cells directly influence the metabolism of fat, maybe more than the other Alpha and Beta receptors the fat cells possess.
This increase in metabolism of fat is why Clenbuterol has often been given to cattle in the past, along with a variety of anabolic steroids, so that the cattle would have more lean meat.
Below are the five main effects of taking Clenbuterol pills:
It is also important to keep in mind that Clenbuterol may work differently in different individuals.
Some people may lose more fat with Clenbuterol, while some might find that they lose more fat with drugs such as Ephedrine, since it reacts with a wider variety of receptors than does Clenbuterol.
However, the important thing to note is that though Clenbuterol works well to stimulate fat loss for most people, there are those non-responders, those who don’t respond well, who do exist.
The half-life of Clenbuterol is about 36 to 48 hours, so there is no need to take more than one dose throughout the day, just once daily is enough.
The last thing to point out concerning the agonistic activity of Clenbuterol, is that it downregulates Beta-2 receptors.
When you use Clenbuterol daily, Beta-2 receptors will regulate, or get used to the activity of Clenbuterol.
This means that Clen’s effect on fat loss will diminish over time. This can be dealt with through a couple of different methods.
The first is to take two weeks or more off of Clen.
Research has shown, however, that using the anti-histamine Ketotifen Fumerate will up-regulate the Beta-2 receptors that Clen down-regulates.
We will talk about this more later, but in about the second or third week of using Clenbuterol, fat loss begins to diminish, though the time frame is different for each person.
This is why it is typically used in bodybuilding cutting cycles for a short period of time.
Then, you may decide to cycle off and use other anabolic steroids to help you bulk up and build muscle. But do not expect to build a lot of muscle during the time that you are taking Clen.
Both men and women can take Clenbuterol HCL to burn fat and get ripped. It is commonly added to steroid cutting stacks or can be used on its own in a Clen-only cycle.
For men, the typical dosage range of this drug is between 40 – 120 mcg per day. Women usually will take between 20 – 60 mcg per day, depending on their bodyweight.
Most clen pills come in a formulation of either 20 or 40 mcg per tablet, though some brands may sell them in 50 or 60 mcg dosages. There are also liquid products, sprays and gels for which you will need to calculate the dosage based on the mcg / mL (i.e. 200 mcg / mL in a 30 mL vial).
Below is a typical dosage chart for men taking Clen to lose weight:
Take all dosages early in the day to prevent your sleep cycle from being interfered with. Drink lots of water and eat well when on this cycle.
You should also be conducting an active workout regimen while on the Clenbuterol diet plan, exercising at least 5 times a week and engaging in both HIIT cardio and strength training.
At the completion of the cycle, it is important to taper your doses as opposed to stopping suddenly. This can prevent any withdrawal symptoms from occuring.
You should then stop taking this drug for a minimum of two weeks so that your tolerance level resets. Some male bodybuilders switch to using an ECA or NYC stack during the off-period of this cutting cycle.
Male steroid users often take Clenbuterol in a cutting stack with other anabolic steroids including trenbolone, testosterone, HGH or Dianabol.
In most cases, it its taken after an anabolic steroid bulking cycle rather than combining it while you are on other steroids like Dianabol, Deca Durabolin, Anadrol or Andriol.
For advanced users, combining Clenbuterol with T3/Cytomel can be very effective. Note that this cycle can result in muscle tissue breakdown and lean mass loss if it is not combined with an effective workout program and high-protein diet.
You want to make sure that your diet is promoting fat loss and leaning out while still preserving muscle size and strength. Clen is only mildly anabolic so you cannot count on it to help you put on muscle like other steroids.
Here are the top 5 most popular Clenbuterol stacks for men:
Women who want to use a Clen cycle will need a smaller dosage to acheive the same effects.
Using dosing guidelines provided for men can result in more side effects, since women tend to be more sensitive to the effects of this sympathomimetic agent.
Beginners can take Clen in a cycle on its own, but the best way for women to take Clenbuterol is in a female cutting stack cycle with other anabolic steroids such as Anavar or Winstrol. Clenbuterol results for women after two weeks can be very impressive when combined with other fat loss agents.
The best Female Clenbuterol Only Cycle Dosage Schedule is as follow:
Is Clenbuterol safe to use for men and women? Millions of people have used this drug safely, but there have also been instances of serious adverse effects and even fatalities.
If you look at the people who experienced harmful side effects, usually they are taking very high dosages of the drug, combining it with other drugs and steroids, or have been taking longer than safe cycles.
A common problem for athletes training with Clenbuterol is excess water loss, resulting in dehydration or your core body temperature increasing too much.
It is important to take precautions when using Clenbuterol to prevent these side effects. For example, consume a lot of water to combat the diuretic effect and avoid doing over-strenuous activity – especially in hot weather.
You should always taper your dosages to guage your individual sentivity as well. Starting at the highest dosage is a recipe for dangerous side effects when taking Clen.
Here is a list of some of the most common side effects from Clenbuterol HCL diet pills:
Longer term side effects can include tachycardia, development of arrhythmias and an increased risk of heart attack or stroke.
This drug must be avoided by anyone who has an increased risk for cardiovascular disease or anyone who has experienced a heart attack or stroke previously.
Sticking to a recommended dosage schedule and consulting with a doctor prior to use are important to reduce your risk of Clenbuterol overdose and other negative effects.
Clenbuterol steroid cycles can be helpful for weight loss, but they need to be used in the right way to ensure you stay safe and to get the best fat burning results.